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Synthesis and benzo-fused benzodiazepines employed as probes of the agonist pharmacophore of benzodiazepine receptorsWEIJIANG ZHANG; KOEHLER, K. F; HARRIS, B et al.Journal of medicinal chemistry (Print). 1994, Vol 37, Num 6, pp 745-757, issn 0022-2623Article

A convenient synthesis of new pyrido[3,2-e][1,4]diazepine-2,5-diones and pyrido[2,3-e][1,4]diazepine-2,5-dionesEL BOUAKHER, Abderrahman; LABORIE, Hélène; AADIL, Mina et al.Tetrahedron letters. 2011, Vol 52, Num 39, issn 0040-4039, 4981, 5077-5080 [5 p.]Article

Copper(I)-Catalyzed Cascade Sulfonimidate to Sulfonamide Rearrangement: Synthesis of Imidazo[1,2-a][1,4]diazepin-7(6H)-oneNAGARAJ, Muthupandi; BOOMINATHAN, Muthusamy; PERUMAL, Devanathan et al.Journal of organic chemistry. 2012, Vol 77, Num 14, pp 6319-6326, issn 0022-3263, 8 p.Article

Pyrrolo[1,2-a]thieno[3,2-f][1,4]diazepines: new 4H and 4H-5,6-dihydro derivativesRAULT, I; RAULT, S; ROBBA, M et al.Heterocycles (Sendai). 1994, Vol 38, Num 4, pp 811-818, issn 0385-5414Article

2,3,4,5-Tetrahydro-1H-pyrido[2,3-b and e][1,4]diazepines as inhibitors of the bacterial enoyl ACP reductase, FabIRAMNAUTH, Jailall; SURMAN, Mathew D; AWREY, Donald E et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 18, pp 5359-5362, issn 0960-894X, 4 p.Article

A novel Smiles rearrangement gives access to the A-ring pyridine isomers of the nevirapine ring systemPROUDFOOT, J. R; PATEL, U. R; CAMPBELL, S. J et al.Journal of organic chemistry. 1993, Vol 58, Num 25, pp 6996-7000, issn 0022-3263Article

An efficient one-pot synthesis, structure, antimicrobial and antioxidant investigations of some novel quinolyldibenzo[b,e][1,4]diazepinonesPARMAR, Narsidas J; BARAD, Hitesh A; PANSURIYA, Bhavesh R et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 11, pp 3816-3821, issn 0960-894X, 6 p.Article

Studies on the chemistry of thieno-anellated O,N- and S,N-containing heterocycles. II: Synthesis of thieno[2,3-b]diazepine derivatives with potential CNS activityERKER, T.Journal of heterocyclic chemistry. 1993, Vol 30, Num 3, pp 807-809, issn 0022-152XArticle

Furo[3,2-e]pyrrolo[1,2-a][1,4]diazepine and derivativesCHEDRU, C; DECROIX, B; MOREL, J et al.Journal of heterocyclic chemistry. 1994, Vol 31, Num 4, pp 1027-1032, issn 0022-152XArticle

Research on nitrogen and sulfur heterocyclic compounds : synthesis of 10H-pyrrolo[1,2-a]thieno[3,4-e][1,4]-diazepin-5(4H)-one and some derivativesDAICH, A; MOREL, J; DECROIX, B et al.Journal of heterocyclic chemistry. 1994, Vol 31, Num 2, pp 341-344, issn 0022-152XArticle

Synthesis of new indeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-diones as potential antitumor agentsINSUASTY, Braulio; OROZCO, Fabian; LIZARAZO, Carolina et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 18, pp 8492-8500, issn 0968-0896, 9 p.Article

The reaction of aromatic α,β-unsaturated ketones with 4,5-diamino-1,6-dihydropyrimidin-6-onesINSUASTY, B; RAMOS, M; QUIROGA, J et al.Journal of heterocyclic chemistry. 1994, Vol 31, Num 1, pp 61-64, issn 0022-152XArticle

Study and characterization of crystalline hydrate/polymorph forms of 5,11-dihydro-11-ethyl-5-methyl-8-2-(1-oxido-4-quinolinyl)ethyl-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepin-6-one by solid-state NMR and solution NMRGONNELLA, N. C; SMOLIGA, John A; CAMPBELL, Scot et al.Journal of pharmaceutical and biomedical analysis. 2010, Vol 51, Num 5, pp 1047-1053, issn 0731-7085, 7 p.Article

Selective [3 + 2] Huisgen Cycloaddition. Synthesis of Trans-Disubstituted Triazolodiazepines from Aza-Baylis-Hillman AdductsDECLERCK, Valérie; TOUPET, Loic; MARTINEZ, Jean et al.Journal of organic chemistry. 2009, Vol 74, Num 5, pp 2004-2007, issn 0022-3263, 4 p.Article

New four-component ugi-type reaction. Synthesis of heterocyclic structures containing a pyrrolo[1,2-a][1,4]diazepine fragmentILYN, Alexey P; TRIFILENKOV, Andrey S; KUZOVKOVA, Julia A et al.Journal of organic chemistry. 2005, Vol 70, Num 4, pp 1478-1481, issn 0022-3263, 4 p.Article

Thienotriazolodiazepines as platelet-activating factor antagonists. Steric limitations for the substituent in position 2WALSER, A; FLYNN, T; MASON, C et al.Journal of medicinal chemistry (Print). 1991, Vol 34, Num 4, pp 1440-1446, issn 0022-2623, 7 p.Article

New synthetic equivalent of nitromalonaldehyde treatable in organic mediaNISHIWAKI, Nagatoshi; OGIHARA, Takuma; TAKAMI, Toshiko et al.Journal of organic chemistry. 2004, Vol 69, Num 24, pp 8382-8386, issn 0022-3263, 5 p.Article

Structural Basis for Inhibitor Specificity in Human Poly(ADP-ribose) Polymerase-3LEHTIÖ, Lari; JEMTH, Ann-Sofie; HELLEDAY, Thomas et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 9, pp 3108-3111, issn 0022-2623, 4 p.Article

A Novel One-Pot Pseudo-Five-Component Synthesis of 4,5,6,7-Tetrahydro-1H-1,4-diazepine-5-carboxamide DerivativesSHAABANI, Ahmad; MALEKI, Ali; MOFAKHAM, Hamid et al.Journal of organic chemistry. 2008, Vol 73, Num 10, pp 3925-3927, issn 0022-3263, 3 p.Article

Synthesis and DNA strand breakage activity of some 1,4-diazepinesMIBU, Nobuko; YUKAWA, Miho; KASHIGE, Nobuhiro et al.Chemical and pharmaceutical bulletin. 2003, Vol 51, Num 1, pp 27-31, issn 0009-2363, 5 p.Article

Silver- and Gold-Mediated Domino Transformation: A Strategy for Synthesizing Benzo[e]indolo[1,2-a]pyrrolo/pyrido[2,1-c][1,4]-diazepine-3,9-dionesYU ZHOU; JIAN LI; XUN JI et al.Journal of organic chemistry. 2011, Vol 76, Num 5, pp 1239-1249, issn 0022-3263, 11 p.Article

Divergent Regioselective Synthesis of 2,5,6,7-Tetrahydro-1H-1, 4-diazepin-2-ones and 5H-1,4-BenzodiazepinesATTANASI, Orazio A; DE CRESCENTINI, Lucia; FAVI, Gianfranco et al.Journal of organic chemistry. 2011, Vol 76, Num 20, pp 8320-8328, issn 0022-3263, 9 p.Article

Ugi multicomponent reaction followed by an intramolecular nucleophilic substitution : Convergent multicomponent synthesis of 1-sulfonyl 1,4-diazepan-5-ones and of their benzo-fused derivativesBANFI, Luca; BASSO, Andrea; GUANTI, Giuseppe et al.Journal of organic chemistry. 2007, Vol 72, Num 6, pp 2151-2160, issn 0022-3263, 10 p.Article

Pyrrolo[3,2-e][1,4]diazepin-2-one Synthesis: A Head-to-Head Comparison of Soluble versus Insoluble SupportsBOUTARD, Nicolas; DUFOUR-GALLANT, Julien; DEAUDELIN, Philippe et al.Journal of organic chemistry. 2011, Vol 76, Num 11, pp 4533-4545, issn 0022-3263, 13 p.Article

Benzothiophene inhibitors of MK2. Part 2: Improvements in kinase selectivity and cell potencyANDERSON, David R; MEYERS, Marvin J; KURUMBAIL, Ravi G et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 16, pp 4882-4884, issn 0960-894X, 3 p.Article

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